CA2113914A1 - Phospholipid derivative and liposome containing it - Google Patents

Phospholipid derivative and liposome containing it

Info

Publication number
CA2113914A1
CA2113914A1 CA002113914A CA2113914A CA2113914A1 CA 2113914 A1 CA2113914 A1 CA 2113914A1 CA 002113914 A CA002113914 A CA 002113914A CA 2113914 A CA2113914 A CA 2113914A CA 2113914 A1 CA2113914 A1 CA 2113914A1
Authority
CA
Canada
Prior art keywords
phospholipid derivative
liposome containing
phospholipid
derivative
moiety
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002113914A
Other languages
French (fr)
Other versions
CA2113914C (en
Inventor
Toshiaki Tagawa
Kaoru Awane
Kazuhiro Nagaike
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsubishi Chemical Corp
Original Assignee
Mitsubishi Kasei Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Kasei Corp filed Critical Mitsubishi Kasei Corp
Publication of CA2113914A1 publication Critical patent/CA2113914A1/en
Application granted granted Critical
Publication of CA2113914C publication Critical patent/CA2113914C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Liposomes
    • A61K9/1271—Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/5537—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom the heteroring containing the structure -C(=O)-N-C(=O)- (both carbon atoms belong to the heteroring)

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A phospholipid derivative of the following formula (I):
CA002113914A 1993-01-22 1994-01-20 Phospholipid derivative and liposome containing it Expired - Fee Related CA2113914C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP02765193A JP3351476B2 (en) 1993-01-22 1993-01-22 Phospholipid derivatives and liposomes containing the same
JP27651/1993 1993-01-22

Publications (2)

Publication Number Publication Date
CA2113914A1 true CA2113914A1 (en) 1994-07-23
CA2113914C CA2113914C (en) 2003-07-29

Family

ID=12226829

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002113914A Expired - Fee Related CA2113914C (en) 1993-01-22 1994-01-20 Phospholipid derivative and liposome containing it

Country Status (6)

Country Link
US (2) US5556948A (en)
EP (1) EP0607978B1 (en)
JP (1) JP3351476B2 (en)
CA (1) CA2113914C (en)
DE (1) DE69421631T2 (en)
ES (1) ES2140473T3 (en)

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