CN102875430A - 莫达非尼多晶型 - Google Patents
莫达非尼多晶型 Download PDFInfo
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- CN102875430A CN102875430A CN2012103955547A CN201210395554A CN102875430A CN 102875430 A CN102875430 A CN 102875430A CN 2012103955547 A CN2012103955547 A CN 2012103955547A CN 201210395554 A CN201210395554 A CN 201210395554A CN 102875430 A CN102875430 A CN 102875430A
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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Abstract
Description
Claims (22)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
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US40206402P | 2002-08-09 | 2002-08-09 | |
US60/402,064 | 2002-08-09 | ||
US10/635,445 | 2003-08-07 | ||
US10/635,445 US6992219B2 (en) | 2002-08-09 | 2003-08-07 | Modafinil polymorphic forms |
Related Parent Applications (1)
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CNB038190850A Division CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
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Publication Number | Publication Date |
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CN102875430A true CN102875430A (zh) | 2013-01-16 |
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CNB038190850A Expired - Fee Related CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
CN201210395545.8A Expired - Fee Related CN102875429B (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
CN2012103955547A Pending CN102875430A (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
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CNB038190850A Expired - Fee Related CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
CN201210395545.8A Expired - Fee Related CN102875429B (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
Country Status (11)
Country | Link |
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US (3) | US6992219B2 (zh) |
EP (2) | EP2402311A1 (zh) |
JP (2) | JP4718177B2 (zh) |
CN (3) | CN100506790C (zh) |
AU (1) | AU2003253128B2 (zh) |
CA (4) | CA2840721C (zh) |
IL (3) | IL166301A (zh) |
MX (1) | MXPA05001506A (zh) |
NZ (1) | NZ537840A (zh) |
WO (1) | WO2004014846A1 (zh) |
ZA (1) | ZA200500411B (zh) |
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US6992219B2 (en) * | 2002-08-09 | 2006-01-31 | Cephalon France | Modafinil polymorphic forms |
FR2849029B1 (fr) * | 2002-12-20 | 2005-03-18 | Lafon Labor | Procede de preparation et formes cristallines des enantiomeres optiques du modafinil. |
MXPA05008088A (es) * | 2003-02-24 | 2005-09-21 | Mallinckrodt Inc | Proceso mejorado para preparar benzhidril tioacetamida. |
AU2003230192A1 (en) * | 2003-03-21 | 2004-10-11 | Hetero Drugs Limited | Novel crystalline forms of aripiprazole |
US20050154052A1 (en) * | 2003-03-24 | 2005-07-14 | Hetero Drugs Limited | Novel crystalline forms of (s)-citalopram oxalate |
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CA2701710C (en) | 2004-07-20 | 2013-08-27 | Warner-Lambert Company Llc | Novel forms of [r-(r*,r*)]-2-(4-fluorophenyl)-.beta.,.delta.-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid calcium salt (2:1) |
US20060235008A1 (en) * | 2004-08-19 | 2006-10-19 | Hetero Drugs Limited | Novel polymorphs of efavirenz |
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DK2056811T3 (en) * | 2006-08-14 | 2018-05-22 | Neurohealing Pharmaceuticals Inc | Modafinil-based treatment for premature ejaculation |
EP2083628A1 (en) | 2006-11-10 | 2009-08-05 | Basf Se | Crystalline modification of fipronil |
UA110598C2 (uk) | 2006-11-10 | 2016-01-25 | Басф Се | Спосіб одержання кристалічної модифікації фіпронілу |
EA017180B1 (ru) | 2006-11-10 | 2012-10-30 | Басф Се | Новая кристаллическая модификация фипронила и ее применение |
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CN101641090B (zh) * | 2006-12-19 | 2012-12-05 | 亚勒斯有限公司 | 莫达非尼在制备治疗多动腿综合征的药物中的应用 |
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FR2923482B1 (fr) * | 2007-11-09 | 2010-01-29 | Servier Lab | Nouvelle forme cristalline vi de l'agomelatine, son procede de preparation et les compositions pharmaceutiques qui la contiennent |
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US9380976B2 (en) | 2013-03-11 | 2016-07-05 | Sync-Think, Inc. | Optical neuroinformatics |
WO2015086489A1 (en) | 2013-12-11 | 2015-06-18 | Merck Sharp & Dohme B.V. | Drug delivery system for delivery of anti-virals |
US10413504B2 (en) | 2013-12-11 | 2019-09-17 | Merck Sharp & Dohme Corp. | Intravaginal ring drug delivery system |
US9616068B2 (en) | 2014-10-27 | 2017-04-11 | Pohela LLC | Animal training using cognitive enhancement |
WO2022056428A1 (en) * | 2020-09-14 | 2022-03-17 | Wellstat Therapeutics Corporation | 2',3'-diacetyluridine substituted with acetoacetyl at the 5' position |
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-
2003
- 2003-08-07 US US10/635,445 patent/US6992219B2/en not_active Expired - Fee Related
- 2003-08-08 CN CNB038190850A patent/CN100506790C/zh not_active Expired - Fee Related
- 2003-08-08 AU AU2003253128A patent/AU2003253128B2/en not_active Ceased
- 2003-08-08 CA CA2840721A patent/CA2840721C/en not_active Expired - Fee Related
- 2003-08-08 WO PCT/IB2003/003215 patent/WO2004014846A1/en active Application Filing
- 2003-08-08 NZ NZ537840A patent/NZ537840A/en not_active IP Right Cessation
- 2003-08-08 JP JP2004527153A patent/JP4718177B2/ja not_active Expired - Fee Related
- 2003-08-08 EP EP11171058A patent/EP2402311A1/en not_active Withdrawn
- 2003-08-08 CN CN201210395545.8A patent/CN102875429B/zh not_active Expired - Fee Related
- 2003-08-08 CA CA2804385A patent/CA2804385A1/en not_active Abandoned
- 2003-08-08 CA CA2494010A patent/CA2494010C/en not_active Expired - Fee Related
- 2003-08-08 MX MXPA05001506A patent/MXPA05001506A/es active IP Right Grant
- 2003-08-08 CN CN2012103955547A patent/CN102875430A/zh active Pending
- 2003-08-08 EP EP03784340A patent/EP1575915A1/en not_active Withdrawn
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- 2005-01-17 ZA ZA2005/00411A patent/ZA200500411B/en unknown
- 2005-10-12 US US11/248,442 patent/US7405323B2/en not_active Expired - Fee Related
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2007
- 2007-12-14 US US11/956,877 patent/US7649020B2/en not_active Expired - Fee Related
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2010
- 2010-10-20 JP JP2010235766A patent/JP5307106B2/ja not_active Expired - Fee Related
- 2010-12-13 IL IL209966A patent/IL209966A/en not_active IP Right Cessation
- 2010-12-13 IL IL209965A patent/IL209965A0/en unknown
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