DE122011000010I1 - N-pyrazol a2a rezeptor agonisten - Google Patents

N-pyrazol a2a rezeptor agonisten

Info

Publication number
DE122011000010I1
DE122011000010I1 DE122011000010C DE122011000010C DE122011000010I1 DE 122011000010 I1 DE122011000010 I1 DE 122011000010I1 DE 122011000010 C DE122011000010 C DE 122011000010C DE 122011000010 C DE122011000010 C DE 122011000010C DE 122011000010 I1 DE122011000010 I1 DE 122011000010I1
Authority
DE
Germany
Prior art keywords
pyrazol
receptor agonists
agonists
receptor
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE122011000010C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gilead Palo Alto Inc
Original Assignee
CV Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by CV Therapeutics Inc filed Critical CV Therapeutics Inc
Publication of DE122011000010I1 publication Critical patent/DE122011000010I1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
DE122011000010C 1999-06-22 2000-06-21 N-pyrazol a2a rezeptor agonisten Pending DE122011000010I1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US09/338,185 US6403567B1 (en) 1999-06-22 1999-06-22 N-pyrazole A2A adenosine receptor agonists
PCT/US2000/040281 WO2000078779A2 (en) 1999-06-22 2000-06-21 N-pyrazole a2a receptor agonists
DE60007127T DE60007127T2 (de) 1999-06-22 2000-06-21 N-pyrazol a2a rezeptor agonisten

Publications (1)

Publication Number Publication Date
DE122011000010I1 true DE122011000010I1 (de) 2011-06-16

Family

ID=23323763

Family Applications (2)

Application Number Title Priority Date Filing Date
DE60007127T Expired - Lifetime DE60007127T2 (de) 1999-06-22 2000-06-21 N-pyrazol a2a rezeptor agonisten
DE122011000010C Pending DE122011000010I1 (de) 1999-06-22 2000-06-21 N-pyrazol a2a rezeptor agonisten

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE60007127T Expired - Lifetime DE60007127T2 (de) 1999-06-22 2000-06-21 N-pyrazol a2a rezeptor agonisten

Country Status (27)

Country Link
US (9) US6403567B1 (de)
EP (1) EP1189916B1 (de)
JP (1) JP4727880B2 (de)
KR (1) KR100463300B1 (de)
CN (1) CN1167709C (de)
AR (1) AR024441A1 (de)
AT (1) ATE256141T1 (de)
AU (1) AU760806B2 (de)
BE (1) BE2011C004I2 (de)
BR (1) BRPI0011856B8 (de)
CA (1) CA2377746C (de)
CY (1) CY2011002I1 (de)
DE (2) DE60007127T2 (de)
DK (1) DK1189916T3 (de)
ES (1) ES2209974T3 (de)
FR (1) FR11C0004I2 (de)
HK (1) HK1044952B (de)
IL (2) IL147198A0 (de)
LU (1) LU91785I2 (de)
MX (1) MXPA01013325A (de)
NO (2) NO322457B1 (de)
NZ (1) NZ516334A (de)
PT (1) PT1189916E (de)
TR (1) TR200200588T2 (de)
TW (1) TWI230161B (de)
WO (1) WO2000078779A2 (de)
ZA (1) ZA200200301B (de)

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CN1358191A (zh) 2002-07-10
US20040038928A1 (en) 2004-02-26
DK1189916T3 (da) 2004-03-22
US8278435B2 (en) 2012-10-02
AR024441A1 (es) 2002-10-02
PT1189916E (pt) 2004-03-31
CY2011002I2 (el) 2012-01-25
CA2377746C (en) 2007-04-10
WO2000078779A2 (en) 2000-12-28
ZA200200301B (en) 2003-11-26
BR0011856B1 (pt) 2014-06-17
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US6642210B1 (en) 2003-11-04
BR0011856A (pt) 2004-02-10
KR20020028910A (ko) 2002-04-17
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US8569260B2 (en) 2013-10-29
JP4727880B2 (ja) 2011-07-20
EP1189916A2 (de) 2002-03-27
US7144872B2 (en) 2006-12-05
NO322457B1 (no) 2006-10-09
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US9045519B2 (en) 2015-06-02
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US20060052332A1 (en) 2006-03-09
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US20130058866A1 (en) 2013-03-07
US20070203090A1 (en) 2007-08-30
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