DE69231522D1 - 1-substituierte-4-amino-1h-imidazo 4,5-c chinoline, zwischenprodukte und arzneimittel - Google Patents

1-substituierte-4-amino-1h-imidazo 4,5-c chinoline, zwischenprodukte und arzneimittel

Info

Publication number
DE69231522D1
DE69231522D1 DE69231522T DE69231522T DE69231522D1 DE 69231522 D1 DE69231522 D1 DE 69231522D1 DE 69231522 T DE69231522 T DE 69231522T DE 69231522 T DE69231522 T DE 69231522T DE 69231522 D1 DE69231522 D1 DE 69231522D1
Authority
DE
Germany
Prior art keywords
products
imidazo
substituted
chinoline
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69231522T
Other languages
English (en)
Other versions
DE69231522T2 (de
Inventor
F Gerster
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
3M Co
Original Assignee
Minnesota Mining and Manufacturing Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Minnesota Mining and Manufacturing Co filed Critical Minnesota Mining and Manufacturing Co
Publication of DE69231522D1 publication Critical patent/DE69231522D1/de
Application granted granted Critical
Publication of DE69231522T2 publication Critical patent/DE69231522T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/052—Imidazole radicals
DE69231522T 1991-09-04 1992-08-26 1-substituierte-4-amino-1h-imidazo 4,5-c chinoline, zwischenprodukte und arzneimittel Expired - Fee Related DE69231522T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/754,610 US5268376A (en) 1991-09-04 1991-09-04 1-substituted 1H-imidazo[4,5-c]quinolin-4-amines
PCT/US1992/007226 WO1993005042A1 (en) 1991-09-04 1992-08-26 1-substituted 1h-imidazo(4,5-c)quinolin-4-amines; intermediate and pharmaceutical compositions

Publications (2)

Publication Number Publication Date
DE69231522D1 true DE69231522D1 (de) 2000-11-23
DE69231522T2 DE69231522T2 (de) 2001-05-17

Family

ID=25035560

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69231522T Expired - Fee Related DE69231522T2 (de) 1991-09-04 1992-08-26 1-substituierte-4-amino-1h-imidazo 4,5-c chinoline, zwischenprodukte und arzneimittel

Country Status (18)

Country Link
US (4) US5268376A (de)
EP (1) EP0603251B1 (de)
JP (1) JP3315983B2 (de)
KR (1) KR100233313B1 (de)
AT (1) ATE197050T1 (de)
AU (1) AU2514792A (de)
CA (1) CA2116782C (de)
CZ (1) CZ281726B6 (de)
DE (1) DE69231522T2 (de)
DK (1) DK0603251T3 (de)
ES (1) ES2150918T3 (de)
HU (4) HU217715B (de)
IL (1) IL102951A (de)
MX (1) MX9205046A (de)
NZ (1) NZ244075A (de)
PH (1) PH30132A (de)
WO (1) WO1993005042A1 (de)
ZA (1) ZA926456B (de)

Families Citing this family (266)

* Cited by examiner, † Cited by third party
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US6894060B2 (en) * 2000-03-30 2005-05-17 3M Innovative Properties Company Method for the treatment of dermal lesions caused by envenomation
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