DE69927936D1 - Präventiva/mittel zur glaukombehandlung - Google Patents

Präventiva/mittel zur glaukombehandlung

Info

Publication number
DE69927936D1
DE69927936D1 DE69927936T DE69927936T DE69927936D1 DE 69927936 D1 DE69927936 D1 DE 69927936D1 DE 69927936 T DE69927936 T DE 69927936T DE 69927936 T DE69927936 T DE 69927936T DE 69927936 D1 DE69927936 D1 DE 69927936D1
Authority
DE
Germany
Prior art keywords
glaucoma
treatment
prophylaxis
agent
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69927936T
Other languages
English (en)
Other versions
DE69927936T2 (de
Inventor
Mitsuyoshi Azuma
Yukuo Yoshida
Mitsunori Waki
Masayoshi Uehata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Senju Pharmaceutical Co Ltd
Mitsubishi Pharma Corp
Original Assignee
Senju Pharmaceutical Co Ltd
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senju Pharmaceutical Co Ltd, Mitsubishi Pharma Corp filed Critical Senju Pharmaceutical Co Ltd
Publication of DE69927936D1 publication Critical patent/DE69927936D1/de
Application granted granted Critical
Publication of DE69927936T2 publication Critical patent/DE69927936T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4409—Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 4, e.g. isoniazid, iproniazid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DE69927936T 1998-08-17 1999-08-13 Präventiva/mittel zur glaukombehandlung Expired - Lifetime DE69927936T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP24776298 1998-08-17
JP24776298 1998-08-17
JP12296099 1999-04-28
JP12296099 1999-04-28
PCT/JP1999/004403 WO2000009162A1 (fr) 1998-08-17 1999-08-13 Medicaments preventifs/curatifs pour le glaucome

Publications (2)

Publication Number Publication Date
DE69927936D1 true DE69927936D1 (de) 2005-12-01
DE69927936T2 DE69927936T2 (de) 2006-06-29

Family

ID=26459997

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69927936T Expired - Lifetime DE69927936T2 (de) 1998-08-17 1999-08-13 Präventiva/mittel zur glaukombehandlung

Country Status (12)

Country Link
US (2) US6673812B1 (de)
EP (3) EP1459743B9 (de)
JP (2) JP3720264B2 (de)
KR (1) KR100616466B1 (de)
CN (2) CN1195547C (de)
AT (3) ATE529102T1 (de)
AU (1) AU5198199A (de)
CA (2) CA2307285C (de)
DE (1) DE69927936T2 (de)
ES (3) ES2247822T3 (de)
HK (3) HK1069120A1 (de)
WO (1) WO2000009162A1 (de)

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Also Published As

Publication number Publication date
HK1030883A1 (en) 2001-05-25
CN1494903A (zh) 2004-05-12
EP1459742A3 (de) 2007-12-26
CA2307285C (en) 2009-03-31
EP1459742A2 (de) 2004-09-22
EP1459742B1 (de) 2011-10-12
ATE527993T1 (de) 2011-10-15
US6673812B1 (en) 2004-01-06
CA2307285A1 (en) 2000-02-24
EP1459743B1 (de) 2011-10-19
ATE529102T1 (de) 2011-11-15
ES2247822T3 (es) 2006-03-01
HK1069120A1 (en) 2005-05-13
ES2372572T3 (es) 2012-01-23
CN1195547C (zh) 2005-04-06
ATE307609T1 (de) 2005-11-15
EP1034793B1 (de) 2005-10-26
AU5198199A (en) 2000-03-06
CN1293878C (zh) 2007-01-10
EP1459742B9 (de) 2012-05-02
CA2635412A1 (en) 2000-02-24
EP1034793A4 (de) 2003-07-09
CN1287494A (zh) 2001-03-14
KR20010015761A (ko) 2001-02-26
EP1459743A8 (de) 2005-02-02
EP1459743A2 (de) 2004-09-22
KR100616466B1 (ko) 2006-08-29
EP1034793A1 (de) 2000-09-13
HK1069121A1 (en) 2005-05-13
EP1459743B9 (de) 2012-08-01
US6649625B2 (en) 2003-11-18
DE69927936T2 (de) 2006-06-29
JP2004277432A (ja) 2004-10-07
US20030125351A1 (en) 2003-07-03
ES2374518T3 (es) 2012-02-17
JP4490748B2 (ja) 2010-06-30
EP1459743A3 (de) 2007-12-26
WO2000009162A1 (fr) 2000-02-24
JP3720264B2 (ja) 2005-11-24
CA2635412C (en) 2011-06-21

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